Jacobio Pharmaceuticals Patent on Solid Forms of Compound I or Salts Thereof
Summary
USPTO published Jacobio Pharmaceuticals' patent application (US20260098039A1) for solid forms of Compound I, a potential cancer therapeutic compound, and its salts. The patent covers novel solid forms, preparation methods, pharmaceutical compositions, and therapeutic uses. The application was filed August 16, 2023, and published April 9, 2026.
What changed
USPTO published Jacobio Pharmaceuticals' patent application for solid forms of Compound I, a heterocyclic compound designated as (S)-5-((1-(3-(5-methyl-3-(trifluoromethyl)-8,9-dihydropyrido[3′,2′:4,5]pyrrolo[1,2-a]pyrazin-7(6H)-yl)-3-oxopropoxy)propan-2-yl)oxy)-4-(trifluoromethyl)pyridazin-3(2H)-one, along with its salts. The patent covers preparation methods and pharmaceutical compositions containing the compound.\n\nPharmaceutical and biotech companies developing cancer therapeutics should review this patent for potential freedom-to-operate concerns and assess whether licensing or design-around strategies may be needed. Researchers and investors may find licensing or collaboration opportunities with Jacobio Pharmaceuticals.
What to do next
- Monitor for updates on patent prosecution status
- Assess freedom-to-operate if developing related cancer therapeutics
- Review licensing opportunities if interested in the patented compound
Archived snapshot
Apr 9, 2026GovPing captured this document from the original source. If the source has since changed or been removed, this is the text as it existed at that time.
SOLID FORMS OF COMPOUND I OR SALTS THEREOF
Application US20260098039A1 Kind: A1 Apr 09, 2026
Assignee
Jacobio Pharmaceuticals Co., Ltd.
Inventors
Haijun LI, Mingming CHEN, Di KANG, Chaojie DANG, Amin LI, Yanping WANG, Wei LONG
Abstract
The present invention relates to novel forms of Compound I, preparation thereof, pharmaceutical composition containing the same and use thereof, wherein, the compound is (S)-5-((1-(3-(5-methyl-3-(trifluoromethyl)-8,9-dihydropyrido[3′,2′:4,5]pyrrolo[1,2-a]pyrazin-7(6H)-yl)-3-oxopropoxy)propan-2-yl)oxy)-4-(trifluoromethyl)pyridazin-3(2H)-one.
CPC Classifications
C07D 471/14 A61K 31/501 A61P 35/00
Filing Date
2023-08-16
Application No.
19104027
Named provisions
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