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Crystalline Nitrogen-Containing Heterocyclic Compound Patent Application

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Published March 25th, 2026
Detected April 2nd, 2026
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Summary

The European Patent Office published patent application EP4480952A1 filed by Shanghai Pharmaceuticals Holding Co., Ltd. for a crystalline form of a nitrogen-containing heterocyclic compound with anti-cancer applications. The application covers the compound's chemical structure, preparation methods, and therapeutic uses under IPC classification C07D471/04.

What changed

The EPO published international patent application EP4480952A1 designating 44 contracting states (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR). The patent protects a crystalline heterocyclic compound classified under C07D471/04 and C07D487/04 with pharmaceutical composition claims targeting cancer (A61P35/00). Inventors include GONG Wanchun, LI Di, LI Ruipeng, DUAN Lingjun, XIA Guangxin, and KE Ying.

This is a standard patent publication with no immediate regulatory obligations. Pharmaceutical companies developing similar heterocyclic compounds should conduct freedom-to-operate analyses to assess potential infringement risks. Patent prosecution will continue through the EPO examination process, with applicants able to validate the patent in any combination of designated contracting states upon grant.

Source document (simplified)

← EPO Patent Bulletin

CRYSTALLINE FORM OF NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF

Publication EP4480952A1 Kind: A1 Mar 25, 2026

Applicants

Shanghai Pharmaceuticals Holding Co., Ltd.

Inventors

GONG, Wanchun, LI, Di, LI, Ruipeng, DUAN, Lingjun, XIA, Guangxin, KE, Ying

IPC Classifications

C07D 471/04 20060101AFI20260219BHEP C07D 487/04 20060101ALI20260219BHEP A61K 31/519 20060101ALI20260219BHEP A61P 35/00 20060101ALI20260219BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR

View original document →

Classification

Agency
EPO
Published
March 25th, 2026
Instrument
Notice
Legal weight
Non-binding
Stage
Final
Change scope
Minor
Document ID
EP4480952A1

Who this affects

Applies to
Pharmaceutical companies Drug manufacturers
Industry sector
3254 Pharmaceutical Manufacturing
Activity scope
Patent Filing Pharmaceutical Compound Protection
Geographic scope
EP EP

Taxonomy

Primary area
Intellectual Property
Operational domain
Legal
Topics
Pharmaceuticals Healthcare

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