Changeflow GovPing Pharma & Drug Safety Novel Heterocyclic Compounds Patent Application
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Novel Heterocyclic Compounds Patent Application

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Published April 2nd, 2026
Detected April 2nd, 2026
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Summary

The USPTO published patent application US20260092073A1 by Hoffmann-La Roche Inc. for novel heterocyclic compounds with general formula I, including compositions and methods of use. The application (Filing Date: 2025-10-15) covers compounds where R1, R2, R9, A1, Rx and Ry define specific substituents. Inventors include David BON, Lea Aurelie BOUCHE, Wolfgang GUBA, and others. CPC Classification: C07D 498/04.

What changed

Hoffmann-La Roche Inc. filed patent application US20260092073A1 for novel heterocyclic compounds having general formula I, covering compositions containing these compounds and methods of using them. The application was published April 2, 2026 with filing date October 15, 2025. Nine inventors are named including David BON, Lea Aurelie BOUCHE, and Wolfgang GUBA. CPC Classification C07D 498/04 indicates fused heterocyclic systems with bridgehead nitrogen atoms.\n\nPharmaceutical companies and drug manufacturers should review the patent claims to assess freedom-to-operate for any heterocyclic compound development programs. While patent applications do not create immediate compliance obligations, monitoring issued patents from competitors is essential for R&D planning. No deadlines or penalties apply to this publication.

Source document (simplified)

← USPTO Patent Applications

NOVEL COMPOUNDS

Application US20260092073A1 Kind: A1 Apr 02, 2026

Assignee

Hoffmann-La Roche Inc.

Inventors

David BON, Lea Aurelie BOUCHE, Wolfgang GUBA, Georg JAESCHKE, Stefanie Katharina MESCH, Angélique PATINY-ADAM, Christian SCHNIDER, Jonathan Martin SHANNON, Sandra STEINER, Andreas Michael TOSSTORFF

Abstract

The invention relates to novel compounds having the general formula I wherein R1, R2, R9, A1, Rx and Ry are as described herein, composition including the compounds and methods of using the compounds.

CPC Classifications

C07D 498/04

Filing Date

2025-10-15

Application No.

19358658

View original document →

Classification

Agency
USPTO
Published
April 2nd, 2026
Instrument
Notice
Legal weight
Non-binding
Stage
Final
Change scope
Minor
Document ID
US20260092073A1
Docket
US20260092073A1

Who this affects

Applies to
Pharmaceutical companies Drug manufacturers
Industry sector
3254 Pharmaceutical Manufacturing
Activity scope
Patent Filing
Geographic scope
United States US

Taxonomy

Primary area
Intellectual Property
Operational domain
Legal
Topics
Pharmaceuticals Healthcare

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