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Pharmaceutical formulations

Grant US12594243B2 Kind: B2 Apr 07, 2026

Assignee

THERACOSBIO, LLC

Inventors

Feng Wang, Ankit Shrivastava, Rina Shah, Brian Seed, Vinay Patil, Michael J. Hadd, Fuxia Dong, Vipan Dhall, Chunfeng Dai, Joseph Ho-Lun Chau, Qiuhua Cai

Abstract

The pharmacokinetic profile of the SGLT2 inhibitor bexagliflozin can be improved by formulating it as an extended release tablet. Compared with standard immediate-release dosage forms these tablets can permit a lower peak plasma concentration, Cmax, while maintaining plasma concentrations at therapeutic levels for a desired period. This can be used, for instance, to administer lower doses while still providing the same pharmacological effect.

CPC Classifications

A61K 9/2013 A61K 9/006 A61K 9/2054 A61K 9/284 A61K 31/70

Filing Date

2023-11-03

Application No.

18501714

Claims

7