← USPTO Patent Grants

Spiromacrocyclic orexin 2 receptor agonists

Grant US12590106B2 Kind: B2 Mar 31, 2026

Assignee

H. Lundbeck A/S

Inventors

Karsten Juhl, Wanwan Yu, Thomas Leegaard Andersen, Erhad Ascic, Michael Baek, Gitte Kobberøe Mikkelsen, Andreas Michael Arnold, Anders Højgaard Hansen, Petra Lindovská, Henrik Juhani Keränen, Ferran Planas Padrós

Abstract

The present invention relates to novel spiro-macrocyclic compounds of general formula (I) which are Orexin 2 receptor agonists.

CPC Classifications

C07D 498/14 C07D 498/04 C07D 513/04 A61K 31/424 A61K 31/4245 A61K 31/429 A61K 31/437 A61K 31/519

Filing Date

2025-04-30

Application No.

19195185

Claims

18