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Salt form and crystal form of A2A receptor antagonist and preparation method therefor

Grant US12583869B2 Kind: B2 Mar 24, 2026

Assignee

CSTONE PHARMACEUTICAL (SUZHOU) CO., LTD.

Inventors

Kevin X Chen, Kai Zhou, Yanxin Yu, Boyu Hu, Li Zhang, Zhaoguo Chen

Abstract

Provided are a salt form and a crystal form of adenosine A2A receptor antagonist, and preparation method therefor. Also provided is an application of the salt form or crystal form in the preparation of a medicine for A2A receptor-related diseases, the maleate salt in the salt form has a structure of formula (I).

CPC Classifications

C07D 519/00 C07B 2200/13 Y02A 50/30 A61P 35/00 C07C 57/145 C07C 309/04 C07C 309/30

Filing Date

2020-03-27

Application No.

17442688

Claims

4