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1,2,4-triazolone derivative as DHODH inhibitor, and preparation method therefor and use thereof

Grant US12577250B2 Kind: B2 Mar 17, 2026

Assignee

WIGEN BIOMEDICINE TECHNOLOGY (SHANGHAI) CO., LTD.

Inventors

Yuli Xie, Houxing Fan, Lihui Qian

Abstract

The present invention relates to a 1,2,4-triazolone derivative as a DHODH inhibitor, a preparation method therefor and use thereof. Specifically, the present invention relates to a compound of general formula (1), a preparation method therefor, and use of the compound of general formula (1) and an isomer, a crystalline form, a pharmaceutically acceptable salt, a hydrate or a solvate thereof as a DHODH inhibitor in the treatment of DHODH-related diseases.

CPC Classifications

A61K 31/4196 A61K 31/437 A61K 31/444 A61K 31/55 C07D 471/04 C07D 487/04 A61P 35/00

Filing Date

2022-07-05

Application No.

18288803

Claims

6