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Solid forms of APOL1 inhibitor and methods of using same

Grant US12577233B2 Kind: B2 Mar 17, 2026

Assignee

Vertex Pharmaceuticals Incorporated

Inventors

Kevin James Gagnon, Jicong Li, Ales Medek, Jack Raphael Minchom, Yi Shi, Muna Shrestha, Faith Witkos

Abstract

The disclosure provides novel solid state forms of Compound I selected from ethanol solvate Form A, ethanol solvate Form B, citric acid cocrystal Form A, and Form B, compositions comprising the same, and methods of making and using the same, including use in treating APOL1 mediated kidney disease. (I).

CPC Classifications

C07D 403/12 C07B 2200/13

Filing Date

2021-06-11

Application No.

18001371

Claims

28