2H-BENZOTRIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME
Application
US20260098034A1
Kind: A1
Apr 09, 2026
Inventors
Peng WANG, Yuqing ZHAO, Yan ZHOU, Lirong ZHANG, Jie ZHOU, Xin ZHOU
Abstract
The invention discloses a benzisothiazole compound as well as a pharmaceutical composition and application thereof, belongs to the technical field of medicines, and particularly relates to a 2H-benzotriazole substituted benzisothiazole compound with a novel structure as shown in a formula (I), a pharmaceutical composition containing the compound and application of the compound in preparation of medicines for treating and/or preventing premature ejaculation. Through in-vivo activity test research, the compound has obviously higher anti-premature ejaculation activity than the on-sale drug dapoxetine.
CPC Classifications
C07D 413/14
A61K 31/454
A61K 31/496
A61P 15/00
C07D 417/14
Filing Date
2023-08-23
Application No.
19112922