COMPOUNDS AND COMPOSITIONS AS SMARCA2/4 DEGRADERS AND USES THEREOF
Application
US20260092071A1
Kind: A1
Apr 02, 2026
Inventors
Shaomeng Wang, Lingying Leng, Lin Yang, Wenbin Tu, Liyue Huang, Mi Wang, Wei Jiang, Paul Kirchhoff, Guozhang Xu, Zhenwu Li, Lalgudi Harikrishnan, E. Scott Priestley, Jelena Tosovic, Jeanne Stuckey
Abstract
Described herein are compounds of Formula II and their pharmaceutically acceptable salts, solvates, or stereoisomers, as well as their uses (e.g., as SMARCA2 or SMARCA4 degraders).
CPC Classifications
C07D 487/10
A61K 31/519
A61K 31/527
A61K 31/5377
A61K 31/541
C07D 471/20
C07D 487/04
C07D 487/20
C07D 491/20
C07D 519/00
Filing Date
2023-09-22
Application No.
19112750