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INHIBITORS FOR PROTEIN N-TERMINAL METHYLTRANSFERASE AND USES THEREOF

Application US20260078147A1 Kind: A1 Mar 19, 2026

Inventors

Rong HUANG, Dongxing Chen, Guangping Dong

Abstract

The present invention relates to series of peptidomimetic compounds as an inhibitor targeting protein N-terminal methyltransferase pharmacological pathway. Pharmaceutical compositions of those compounds and methods of using them in the treatment of diseases caused by abnormal protein methyltransferase pathway, including cancer, inflammation, neurodegenerative and cardiovascular diseases, are within the scope of this disclosure.

CPC Classifications

C07K 7/08 C07K 7/06 A61K 38/00 A61P 9/00 A61P 25/28 A61P 29/00 A61P 35/00 C07K 5/0823 C07K 5/1024

Filing Date

2025-10-20

Application No.

19363450