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Macrocyclic Compounds as RAS Inhibitors

Application US20260078134A1 Kind: A1 Mar 19, 2026

Assignee

BeOne Medicines I GmbH

Inventors

Jing Li, Yian Guo, Sanjia Xu, Zhiwei Wang

Abstract

Provided herein are compounds having the following structure: or pharmaceutically acceptable salts, hydrates, or solvates thereof, wherein the substituents are as defined herein, their pharmaceutical compositions and uses for modulating the activity of multiple RAS mutants.

CPC Classifications

C07D 513/22 A61K 31/504 A61K 31/5377 A61K 31/5383 A61K 31/5386 A61K 31/551 C07D 519/00

Filing Date

2025-09-18

Application No.

19332430