NAMPT MODULATORS, PREPARATIONS, AND USES THEREOF
Application
US20260078130A1
Kind: A1
Mar 19, 2026
Inventors
Xiaoqing WANG, Weijie HOU, Ming JIANG, Shaoqiang YANG, Tao SHENG, Guangxin LI, Jie LU, Yingtao LIU, Yu CHEN, Lianzhu LIU, Yimin JIANG, Yanping XU, Zhiyuan ZHANG
Abstract
This disclosure provides compounds of Formula 1 or 8, compositions comprising the same, and methods of using the same, including uses in modulating NAMPT and treating various diseases and conditions that are responsive to NAMPT activation.
CPC Classifications
C07D 487/10
A61K 31/4035
A61K 31/4155
A61K 31/416
A61K 31/4184
A61K 31/4192
A61K 31/422
A61K 31/423
A61K 31/4245
A61K 31/427
A61K 31/428
A61K 31/429
A61K 31/433
A61K 31/437
A61K 31/4439
A61K 31/444
A61K 31/454
A61K 31/4704
A61K 31/4725
A61K 31/4985
A61K 31/501
A61K 31/506
A61K 31/517
A61K 31/5377
A61K 31/538
C07B 59/002
C07D 209/46
C07D 209/48
C07D 215/227
C07D 217/24
C07D 231/56
C07D 265/36
C07D 401/06
C07D 401/12
C07D 401/14
C07D 403/04
C07D 403/06
C07D 403/12
C07D 403/14
C07D 405/14
C07D 413/06
C07D 413/14
C07D 417/06
C07D 417/14
C07D 471/04
C07D 487/04
C07D 491/107
C07D 498/04
C07D 513/04
C07B 2200/05
Filing Date
2023-09-22
Application No.
19109179