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Novel Aminocarboxymuconate Semialdehyde Decarboxylase Inhibitors

Application US20260078105A1 Kind: A1 Mar 19, 2026

Inventors

Archana Vijayakumar, Gary Phillips, Eisuke Murakami, G. Mani Subramanian

Abstract

Disclosed herein are inhibitors of aminocarboxymuconate semialdehyde decarboxylase (ACMSD), pharmaceutical compositions and methods for using these compounds to treat or prevent one or more ACMSD-related diseases such as, for example, muscle structure disorders, neuronal activation disorders, muscle fatigue disorders, muscle mass disorders, beta oxidation diseases, metabolic diseases, cancer, vascular diseases, ocular vascular diseases, muscular eye diseases, liver diseases, inflammatory diseases or renal diseases.

CPC Classifications

C07D 401/12 A61K 31/4418 A61K 31/4439 A61K 31/444 A61K 31/496 A61K 31/506 A61K 31/513 A61K 31/53 C07D 213/85 C07D 239/56 C07D 401/14 C07D 403/12

Filing Date

2024-10-11

Application No.

18913029