PYRAZOLO[4,3-F]QUINAZOLINE DERIVATIVES AS MODULATORS OF G12D MUTANT KRAS USEFUL FOR THE TREATMENT OF CANCER
Publication
EP4709729A1
Kind: A1
Mar 18, 2026
Applicants
Jazz Pharmaceuticals Ireland Ltd.
Inventors
JACKSON, Paula, AYLOTT, Helen Elizabeth, JONES, Clifford D, BHAMRA, Inder, RYAN, James, LENG, Daniel J, HO, Kelvin
IPC Classifications
C07D 487/04 20060101AFI20241122BHEP
C07D 519/00 20060101ALI20241122BHEP
A61K 31/517 20060101ALI20241122BHEP
A61P 35/00 20060101ALI20241122BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR