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THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS AND USES THEREOF

Publication EP4630119A1 Kind: A1 Mar 18, 2026

Applicants

GlaxoSmithKline Intellectual Property (No.4) Limited, Ideaya Biosciences, Inc.

Inventors

BOTYANSZKI, Janos, DUFFY, Kevin, NEILAN, Claire L., FISCHER, Marcus Michael, CHOI, Young Eun

IPC Classifications

A61P 35/00 20060101AFI20240614BHEP C07D 417/14 20060101ALI20240614BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR