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N-PHENYL-PYRAZOLO[1,5-A]PYRIDINE-3-CARBOXAMIDE DERIVATIVES AS WILD TYPE C-KIT KINASE INHIBITORS FOR THE TREATMENT OF URTICARIA

Publication EP4626884A1 Kind: A1 Mar 11, 2026

Applicants

Blueprint Medicines Corporation

Inventors

BRUBAKER, Jason, D., DAI, Yinghui, DINEEN, Thomas, A., DU, Guangyan, FANG, Cheng, HAIDLE, Andrew, Marc, KIM, Joseph, L., PEROLA, Emanuele, SAMARAKOON, Thiwanka, WILSON, Douglas

IPC Classifications

C07D 471/04 20060101AFI20240607BHEP A61K 31/437 20060101ALI20240607BHEP A61P 3/10 20060101ALI20240607BHEP A61P 9/12 20060101ALI20240607BHEP A61P 11/00 20060101ALI20240607BHEP A61P 11/06 20060101ALI20240607BHEP A61P 17/00 20060101ALI20240607BHEP A61P 17/06 20060101ALI20240607BHEP A61P 25/00 20060101ALI20240607BHEP A61P 25/28 20060101ALI20240607BHEP A61P 29/00 20060101ALI20240607BHEP A61P 35/00 20060101ALI20240607BHEP A61P 35/02 20060101ALI20240607BHEP A61P 37/00 20060101ALI20240607BHEP A61P 37/02 20060101ALI20240607BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR