PREPARATION OF FUSED AZOLE DERIVATIVES AS NOVEL DIACYLGLYCERIDE O-ACYLTRANSFERASE 2 INHIBITORS
Publication
EP4626881A1
Kind: A1
Mar 11, 2026
Applicants
Merck Sharp & Dohme LLC
Inventors
LIM, Yeon-Hee, HUGELSHOFER, Cedric L., ROANE, James P., SHOCKLEY, Samantha E.
IPC Classifications
C07D 409/14 20060101AFI20240607BHEP
C07D 413/12 20060101ALI20240607BHEP
C07D 413/14 20060101ALI20240607BHEP
C07D 417/14 20060101ALI20240607BHEP
C07D 471/04 20060101ALI20240607BHEP
C07D 487/04 20060101ALI20240607BHEP
C07D 498/04 20060101ALI20240607BHEP
C07D 513/04 20060101ALI20240607BHEP
A61P 3/00 20060101ALI20240607BHEP
A61P 9/00 20060101ALI20240607BHEP
A61P 25/00 20060101ALI20240607BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR