CYCLIC PYRAZOLE DIAMIDE IRE1/XBP1S ACTIVATORS
Publication
EP4626865A1
Kind: A1
Mar 11, 2026
Applicants
Protego Biopharma, Inc.
Inventors
LABAUDINIERE, Richard F., TAIT, Bradley Dean, QIU, Huang, PETRASSI, Hank Michael James, QIN, Bo
IPC Classifications
C07D 231/40 20060101AFI20250618BHEP
C07D 401/06 20060101ALI20250618BHEP
C07D 401/12 20060101ALI20250618BHEP
C07D 401/14 20060101ALI20250618BHEP
C07D 403/06 20060101ALI20250618BHEP
C07D 403/12 20060101ALI20250618BHEP
C07D 403/14 20060101ALI20250618BHEP
C07D 405/12 20060101ALI20250618BHEP
C07D 405/14 20060101ALI20250618BHEP
C07D 413/12 20060101ALI20250618BHEP
C07D 413/14 20060101ALI20250618BHEP
A61P 1/16 20060101ALI20250618BHEP
A61P 3/10 20060101ALI20250618BHEP
A61P 9/10 20060101ALI20250618BHEP
A61P 25/02 20060101ALI20250618BHEP
A61P 25/08 20060101ALI20250618BHEP
A61P 25/14 20060101ALI20250618BHEP
A61P 25/16 20060101ALI20250618BHEP
A61P 25/28 20060101ALI20250618BHEP
A61P 27/02 20060101ALI20250618BHEP
A61K 31/415 20060101ALI20250618BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR