LINEAR HETEROARYL DIAMIDE IRE1/XBP1S ACTIVATORS
Publication
EP4626864A1
Kind: A1
Mar 11, 2026
Applicants
Protego Biopharma, Inc.
Inventors
LABAUDINIERE, Richard F., TAIT, Bradley Dean, QIU, Huang, PETRASSI, Hank Michael James, QIN, Bo
IPC Classifications
C07D 231/40 20060101AFI20250623BHEP
C07D 285/08 20060101ALI20250623BHEP
C07D 401/12 20060101ALI20250623BHEP
C07D 401/14 20060101ALI20250623BHEP
C07D 403/12 20060101ALI20250623BHEP
C07D 405/12 20060101ALI20250623BHEP
C07D 405/14 20060101ALI20250623BHEP
C07D 471/04 20060101ALI20250623BHEP
C07D 487/04 20060101ALI20250623BHEP
C07D 491/056 20060101ALI20250623BHEP
A61K 31/415 20060101ALI20250623BHEP
A61K 31/433 20060101ALI20250623BHEP
A61K 31/4355 20060101ALI20250623BHEP
A61K 31/437 20060101ALI20250623BHEP
A61K 31/4439 20060101ALI20250623BHEP
A61K 31/497 20060101ALI20250623BHEP
A61K 31/506 20060101ALI20250623BHEP
A61P 1/00 20060101ALI20250623BHEP
A61P 1/16 20060101ALI20250623BHEP
A61P 3/10 20060101ALI20250623BHEP
A61P 9/00 20060101ALI20250623BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR