2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1H)-ONE DERIVATIVES DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER
Publication
EP4612148A1
Kind: A1
Mar 18, 2026
Applicants
Cancer Research Technology Limited
Inventors
WARING, Michael J., STEWART, Hannah L., MARTIN, Mathew P., AL-KHAWALDEH, Islam H., HERBERT, Jack T., HOWARD, Steven, TWIGG, David Geoffrey, LIEBESCHUETZ, John Walter, ST. DENIS, Jeffrey David
IPC Classifications
C07D 471/04 20060101AFI20240510BHEP
C07D 487/04 20060101ALI20240510BHEP
A61P 35/00 20060101ALI20240510BHEP
A61P 35/02 20060101ALI20240510BHEP
A61P 35/04 20060101ALI20240510BHEP
A61K 31/519 20060101ALI20240510BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR