HETEROCYCLIC INHIBITORS OF KRAS G12C MUTANT PROTEINS AND USES THEREOF
Publication
EP4598917A1
Kind: A1
Mar 18, 2026
Applicants
Amgen Inc.
Inventors
LANMAN, Brian A., BOOKER, Shon, BUTLER, John R., GLIBSTRUP, Emil, HUANG, David, HUSEMOEN, Birgitte, KALLER, Matthew R., KOHN, Todd J., LETH-PETERSEN, Sebastian, LOPEZ, Patricia, LIU, Qingyian, MA, Vu Van, MANONI, Francesco, PEIRO CADAHIA, Jorge, PICKRELL, Alexander J., RAST, Slavko, TAMAYO, Nuria A., WANG, Hui-Ling, ZHANG, Wenhan, ZHU, Kai, BANERJEE, Abhisek
IPC Classifications
C07D 401/14 20060101AFI20240412BHEP
C07D 403/14 20060101ALI20240412BHEP
C07D 405/14 20060101ALI20240412BHEP
C07D 417/14 20060101ALI20240412BHEP
A61P 35/00 20060101ALI20240412BHEP
A61K 31/506 20060101ALI20240412BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR