← EPO Patent Bulletin

SUBSTITUTED HETEROCYCLIC COMPOUNDS AND THERAPEUTIC USES THEREOF

Publication EP4509122A2 Kind: A2 Mar 18, 2026

Applicants

Bayer Aktiengesellschaft, The Broad Institute, Inc., Dana-Farber Cancer Institute, Inc.

Inventors

SCHULZE, Volker, MENGEL, Anne, FARIA ALVARES DE LEMOS, Adelaide, Clara, CHRISTIAN, Sven, BÖMER, Ulf, HILLIG, Roman, LECHNER, Christian, MORTIER, Jérémie, Xavier, G., KAULFUSS, Stefan, CORSELLO, Steven, HANDING, Katarzyna, MADEC, Amael, FURST, Laura, SHEKHAR, Mrinal, BERGER, Markus, RUPAIMOOLE, Rajesha, LIENAU, Philip, ORSI, Douglas, MCKINNEY, David, BRZEZINKA, Krzysztof

IPC Classifications

C07D 471/04 20060101AFI20250317BHEP C07D 487/04 20060101ALI20250317BHEP A61P 35/00 20060101ALI20250317BHEP A61K 31/437 20060101ALI20250317BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR