PYRAZOLE MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF
Publication
EP4493557A1
Kind: A1
Mar 18, 2026
Applicants
Insilico Medicine IP Limited
Inventors
DING, Xiao, REN, Feng, WANG, Yazhou, ZHENG, Min
IPC Classifications
C07D 405/14 20060101AFI20260211BHEP
C07D 405/04 20060101ALI20260211BHEP
C07D 405/06 20060101ALI20260211BHEP
C07D 405/08 20060101ALI20260211BHEP
C07D 403/04 20060101ALI20260211BHEP
C07D 231/14 20060101ALI20260211BHEP
C07D 401/04 20060101ALI20260211BHEP
C07D 401/06 20060101ALI20260211BHEP
C07D 413/06 20060101ALI20260211BHEP
A61K 31/4155 20060101ALI20260211BHEP
A61P 35/00 20060101ALI20260211BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR