← EPO Patent Bulletin

NON-AROMATIC CYCLIC-PYRIMIDINE ANALOGS AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS

Publication EP4490148A2 Kind: A2 Mar 18, 2026

Applicants

Merck Sharp & Dohme LLC

Inventors

WALSH, Shawn P., TAN, Zheng, TONG, Ling, SLUTSKYY, Yuriy, NEELAMKAVIL, Santhosh Francis, LIU, Weiguo, DONOFRIO, Anthony

IPC Classifications

C07D 239/24 20060101AFI20240920BHEP A61K 31/505 20060101ALI20240920BHEP A61P 35/00 20060101ALI20240920BHEP A61P 25/16 20060101ALI20240920BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, ME, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR