N-(PHENYL)-5-(HETEROARYL)-1H-PYRAZOL-3-AMINE DERIVATIVES AS TNIK INHIBITORS FOR USE IN THE TREATMENT OF CANCER
Publication
EP4477271A2
Kind: A2
Mar 18, 2026
Applicants
Korea Research Institute of Chemical Technology, Industry-Academic Cooperation Foundation, Yonsei University
Inventors
CHANG, Sung Youn, LEE, Hyuk, KIM, Ki Young, KIM, Bum Tae, KIM, Sung Soo, KIM, Seong Hwan, LIM, Hwan Jung, HEO, Jung Nyoung, SHIN, Sang Joon, PARK, Sang Youn
IPC Classifications
C07D 231/38 20060101AFI20251209BHEP
C07D 401/04 20060101ALI20251209BHEP
C07D 401/14 20060101ALI20251209BHEP
C07D 403/04 20060101ALI20251209BHEP
C07D 403/10 20060101ALI20251209BHEP
C07D 403/12 20060101ALI20251209BHEP
C07D 403/14 20060101ALI20251209BHEP
C07D 409/04 20060101ALI20251209BHEP
C07D 413/10 20060101ALI20251209BHEP
C07D 413/12 20060101ALI20251209BHEP
C07D 417/04 20060101ALI20251209BHEP
A61K 31/415 20060101ALI20251209BHEP
A61K 31/4155 20060101ALI20251209BHEP
A61K 31/4178 20060101ALI20251209BHEP
A61K 31/4439 20060101ALI20251209BHEP
A61P 35/00 20060101ALI20251209BHEP
A61P 35/02 20060101ALI20251209BHEP
A61P 35/04 20060101ALI20251209BHEP
C07D 401/10 20060101ALN20251209BHEP
A61K 31/427 20060101ALN20251209BHEP
A61K 31/454 20060101ALN20251209BHEP
A61K 31/4745 20060101ALN20251209BHEP
A61K 31/496 20060101ALN20251209BHEP
A61K 31/5377 20060101ALN20251209BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR