N-(2-OXO-3,4-DIHYDRO-1H-QUINOLIN-6-YL)-PYRIDINE-4-CARBOXAMIDE DERIVATIVES AS ALDH INHIBITORS FOR THE TREATMENT OF CANCER
Publication
EP4326696A1
Kind: A1
Mar 25, 2026
Applicants
Kayothera Inc., The Trustees of Princeton University
Inventors
ESPOSITO, Mark, PROUDFOOT, John, KANG, Yibin, PIWINSKI, John
IPC Classifications
C07D 215/38 20060101AFI20251211BHEP
C07D 221/04 20060101ALI20251211BHEP
C07D 401/12 20060101ALI20251211BHEP
C07D 405/12 20060101ALI20251211BHEP
C07D 405/14 20060101ALI20251211BHEP
C07D 413/12 20060101ALI20251211BHEP
C07D 417/12 20060101ALI20251211BHEP
C07D 471/04 20060101ALI20251211BHEP
C07D 491/048 20060101ALI20251211BHEP
C07D 498/04 20060101ALI20251211BHEP
C07D 513/04 20060101ALI20251211BHEP
A61K 31/4704 20060101ALI20251211BHEP
A61P 35/00 20060101ALI20251211BHEP
A61P 3/00 20060101ALI20251211BHEP
A61P 3/10 20060101ALI20251211BHEP
A61P 9/12 20060101ALI20251211BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR