← EPO Patent Bulletin

CRYSTALLINE FORMS OF (2R,5S,13AR)-8-HYDROXY-7,9-DIOXO-N-(2,4,6-TRIFLUOROBENZYL)-2,3,4,5,7,9,13,13A-OCTAHYDRO-2,5-METHANOPYRIDO [1',2':4,5]PYRAZINO [2,1-B][1,3]OXAZEPINE-10-CARBOXAMIDE

Publication EP4309736A2 Kind: A2 Mar 18, 2026

Applicants

Gilead Sciences, Inc.

Inventors

CARRA, Ernest A., CHEN, Irene, KEATON, Katie Ann, ZIA, Vahid

IPC Classifications

C07D 498/18 20060101AFI20260206BHEP A61K 31/513 20060101ALI20260206BHEP A61P 31/18 20060101ALI20260206BHEP A61P 43/00 20060101ALI20260206BHEP A61K 45/06 20060101ALI20260206BHEP A61K 31/553 20060101ALI20260206BHEP A61K 31/675 20060101ALI20260206BHEP A61K 31/683 20060101ALI20260206BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR