← EPO Patent Bulletin

TETRAHYDROQUINAZOLINE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS

Publication EP4259608A1 Kind: A1 Mar 18, 2026

Applicants

Merck Sharp & Dohme LLC

Inventors

CONVERSO, Antonella, HUNTER, David N., EL MARROUNI, Abdellatif, ROECKER, Anthony J., SHAW, Anthony W., SHIPE, William D., WANG, Cheng, WANG, Deping, ZHANG, Yunlong

IPC Classifications

C07D 239/80 20060101AFI20240924BHEP C07D 401/06 20060101ALI20240924BHEP C07D 403/06 20060101ALI20240924BHEP A61P 31/18 20060101ALI20240924BHEP A61P 31/12 20060101ALI20240924BHEP A61K 31/517 20060101ALI20240924BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR