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NOVEL 6-6 BICYCLIC AROMATIC RING SUBSTITUTED NUCLEOSIDE ANALOGUES FOR USE AS PRMT5 INHIBITORS

Publication EP4219496A1 Kind: A1 Mar 18, 2026

Applicants

JANSSEN Pharmaceutica NV

Inventors

WU, Tongfei, BREHMER, Dirk, BEKE, Lijs, BOECKX, An, DIELS, Gaston, Stanislas, Marcella, GILISSEN, Ronaldus, Arnodus, Hendrika, Joseph, LAWSON, Edward, Charles, PANDE, Vineet, PARADE, Marcus, Cornelis, Bernardus, Catharina, SCHEPENS, Wim, Bert, Griet, THURING, Johannes, Wilhelmus, John, F., VIELLEVOYE, Marcel, SUN, Weimei, MEERPOEL, Lieven

IPC Classifications

C07D 471/04 20060101AFI20230621BHEP A61K 31/519 20060101ALI20230621BHEP A61K 31/53 20060101ALI20230621BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR