PIPERIDINE-2,6-DIONES AS SMALL MOLECULE DEGRADERS OF HELIOS AND METHODS OF USE
Publication
EP4153175A1
Kind: A1
Mar 18, 2026
Applicants
Dana-Farber Cancer Institute, Inc.
Inventors
GRAY, Nathanael S., FISCHER, Eric S., VERANO, Alyssa, LIU, Hu, ZHANG, Tinghu, JONES, Lyn H., WANG, Eric S., NOWAK, Radoslaw, CHE, Jianwei
IPC Classifications
C07D 401/04 20060101AFI20240429BHEP
C07D 401/14 20060101ALI20240429BHEP
A61K 31/445 20060101ALI20240429BHEP
A61K 31/454 20060101ALI20240429BHEP
A61P 35/02 20060101ALI20240429BHEP
A61P 13/12 20060101ALI20240429BHEP
A61P 19/06 20060101ALI20240429BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR