← EPO Patent Bulletin

MACROCYCLIC PAD4 INHIBITORS USEFUL AS IMMUNOSUPPRESSANT

Publication EP4100405A1 Kind: A1 Mar 18, 2026

Applicants

Bristol-Myers Squibb Company

Inventors

NGU, Khehyong, ANNUNZIATO, Christopher, DUNCIA, John V., GARDNER, Daniel S.

IPC Classifications

C07D 403/14 20060101AFI20210813BHEP C07D 487/04 20060101ALI20210813BHEP C07D 487/08 20060101ALI20210813BHEP A61K 31/437 20060101ALI20210813BHEP A61K 31/439 20060101ALI20210813BHEP A61K 31/445 20060101ALI20210813BHEP A61P 19/00 20060101ALI20210813BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR