← EPO Patent Bulletin

MACROCYCLES WITH HETEROCYCLIC P2' GROUPS AS FACTOR XIA INHIBITORS

Publication EP3988549A1 Kind: A1 Mar 25, 2026

Applicants

Bristol-Myers Squibb Company

Inventors

CORTE, James R., DE LUCCA, Indawati, FANG, Tianan, YANG, Wu, WANG, Yufeng, DILGER, Andrew K., PABBISETTY, Kumar Balashanmuga, EWING, William R., ZHU, Yeheng, WEXLER, Ruth R., PINTO, Donald J.P., ORWAT, Michael J., SMITH, Leon M. II

IPC Classifications

C07D 471/08 20060101AFI20220221BHEP C07D 487/08 20060101ALI20220221BHEP A61K 31/529 20060101ALI20220221BHEP A61P 7/00 20060101ALI20220221BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR