← EPO Patent Bulletin

PHARMACEUTICALLY ACTIVE PYRAZOLO-PYRIDONE MODULATORS OF DCN1/2-MEDIATED CULLIN NEDDYLATION

Publication EP3986893A1 Kind: A1 Mar 18, 2026

Applicants

University Of Kentucky Research Foundation, Memorial Sloan Kettering Cancer Center, St. Jude Children's Research Hospital, Inc.

Inventors

KIM, Hoshin, GUY, Rodney Kiplin, HAMMILL, Jared T., SCOTT, Daniel Charles, SCHULMAN, Benda Arlene, SINGH, Bhuvanesh

IPC Classifications

C07D 471/04 20060101AFI20230606BHEP C07D 519/00 20060101ALI20230606BHEP A61P 25/28 20060101ALI20230606BHEP A61P 31/00 20060101ALI20230606BHEP A61P 35/00 20060101ALI20230606BHEP A61K 31/437 20060101ALI20230606BHEP

Designated States

AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR