SMALL MOLECULE DEGRADERS OF FKBP12 VIA RECRUITMENT OF VON HIPPEL-LINDAU E3 UBIQUITIN LIGASE (VHL) E3 UBIQUITIN LIGASE, AND USES IN DTAG SYSTEMS
Publication
EP3908291A1
Kind: A1
Mar 18, 2026
Applicants
Dana-Farber Cancer Institute, Inc.
Inventors
GRAY, Nathanael S., FERGUSON, Fleur M., NABET, Behnam, BUCKLEY, Dennis L.
IPC Classifications
A61K 47/55 20170101AFI20260211BHEP
A61K 35/17 20150101ALI20260211BHEP
C12N 9/22 20060101ALI20260211BHEP
C07K 14/82 20060101ALI20260211BHEP
A61K 38/00 20060101ALI20260211BHEP
A61P 35/00 20060101ALI20260211BHEP
C12N 9/10 20060101ALI20260211BHEP
C12N 9/90 20060101ALI20260211BHEP
C07K 14/725 20060101ALI20260211BHEP
C12N 5/0783 20100101ALI20260211BHEP
Designated States
AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR